TABLE 7.
IC50s for E. coli DNA gyrase supercoiling
| Compound | Supercoiling IC50 (μM) |
|---|---|
| Norfloxacin | 0.64 |
| Ofloxacin | 1.14 |
| Ciprofloxacin | 0.25 |
| Compound A | 35.5 |
| Compound B | 41.4 |
| Compound C | 30.1 |
| Compound D | 8.57 |
IC50s for E. coli DNA gyrase supercoiling
| Compound | Supercoiling IC50 (μM) |
|---|---|
| Norfloxacin | 0.64 |
| Ofloxacin | 1.14 |
| Ciprofloxacin | 0.25 |
| Compound A | 35.5 |
| Compound B | 41.4 |
| Compound C | 30.1 |
| Compound D | 8.57 |