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. Author manuscript; available in PMC: 2015 Nov 1.
Published in final edited form as: Bioorg Med Chem Lett. 2014 Sep 15;24(21):5098–5101. doi: 10.1016/j.bmcl.2014.08.066

Table 1.

Potency
(EC50)		 Solubility Human
Metabolic
Potential
(T1/2)		 Mouse
Metabolic
Potential
(T1/2)		 Plasma
Stability
(Calc T1/2)
graphic file with name nihms627115t1.jpg 1.68 uM 31.3 uM 64 min 16 min 63.5 min
graphic file with name nihms627115t2.jpg 1.70 uM 31.3 uM 75 min 16 min 49.8 min
graphic file with name nihms627115t3.jpg 1.57 uM 31.3 uM 64 min 15 min 54.0 min
graphic file with name nihms627115t4.jpg 1.05 uM 62.5 uM 64 min 14 min 49.4 min