Table 2.
A list of inhibitory Gi/o-coupled GPCRs that may be presynaptically-expressed and potentially mediate LTD at various synapses throughout the CNS.
Receptor Family | Receptor |
---|---|
Serotonin | 5-HT1a |
5-HT1b | |
5-HT1d | |
5-HT1e | |
5-HT1f | |
5-HT5a | |
Acetylcholine | M2 |
M4 | |
Adenosine | A1 |
A3 | |
Adrenergic | A2a |
A2b | |
A2c | |
Anaphylatoxin | C5a1/CD88 |
Angiotensin | AT1 |
AT2 | |
Apelin | APJ |
Cannabinoid | CB1 |
Chemokine | CCR2 |
CCR10 | |
CXCR4 | |
CX3CR1 | |
Dopamine | D2 |
D3 | |
D4 | |
Galanin | GAL1 |
GAL2 | |
GAL3 | |
Histamine | H3R |
Leukotriene | BLT1 |
BLT2 | |
OXE | |
FPR2/AXE | |
Lysophospholipid | LPA3 |
S1P1 | |
S1P3 | |
S1P5 | |
MCH | MCH1 |
Melatonin | MT1 |
MT2 | |
MT3 | |
Neuropeptides | DOR |
KOR | |
MOR | |
NOR/ORL-1 | |
NPFF1 | |
NPFF2 | |
NPBW1 | |
NPBW2 | |
Orexin | OX2 |
Purinergic | P2Y1 |
P2Y12 | |
P2Y13 | |
Prokineticin | PKR2 |
Prostanoid | EP3 |
DP2 | |
Relaxin | RXFP2 |
RXFP3 | |
RXFP4 | |
Somatostatin | SSTR1 |
SSTR2 | |
SSTR3 | |
SSTR4 | |
SSTR5 | |
Ca2+ Sensing | CaS |
GABA | GABAB |
mGluR | mGluR2 |
mGluR3 | |
mGluR4 | |
mGluR6 | |
mGluR7 | |
mGluR8 |