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. 2014 Oct 27;171(22):4981–5010. doi: 10.1111/bph.12848

Table 8.

Examples of KDM inhibitors

Name KDM specificity/bias Structure Potency (µM) Reference
OG-L002 KDM1A Inline graphic 0.02 (Liang et al., 2013)
NCL-1 KDM1A Inline graphic 1.6 (Ogasawara et al., 2011)
Daminozide KDM2/7 Inline graphic 1.5–2.1 (Rose et al., 2012)
PBIT KDM5B Inline graphic 3 (Sayegh et al., 2013)
GSK-J1 KDM6A/B Inline graphic 5 (Kruidenier et al., 2012)