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| CYP enzyme | substrate | 1 IC50 (μM) | 2 IC50 (μM) | 3 IC50 (μM) | 4 IC50 (μM) | 5 IC50 (μM) |
|---|---|---|---|---|---|---|
| 1A2 | tacrin | 8.6 | 3.7 | >20 | >20 | >2.5 |
| 2B6 | bupropion | >20 | >20 | >20 | >20 | >2.5 |
| 2C8 | amodiaquine | >20 | >20 | >20 | >20 | >2.5 |
| 2C9 | diclofenac | 19 | 8.8 | >20 | >20 | >2.5 |
| 2C19 | (S)-mephentoin | 6.5 | 7. 9 | >20 | >20 | >2.5 |
| 2D6 | dextromethophan | >20 | >20 | >20 | >20 | >2.5 |
| 3A4 | midazolam | >20 | >20 | >20 | >20 | >2.5 |
| 3A4 | testosterone | >20 | >20 | >20 | >20 | >2.5 |
