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. 2015 Jan 1;5(1):23–42. doi: 10.7150/thno.10202

Table 2.

Application of aptamer-drug conjugations as cancer-targeted therapeutics

Aptamer Target Drug Cancer Research Group
DNA aptamer CCRF-CEM cell DOX T-cell ALL Tan et al. 2009 100
DNA aptamer LH86 cell DOX Human hepatocellular carcinoma Tan et al. 2012 52
DNA aptamer MUC1 protein DOX Lung cancer and breast cancer Yang et al. 2012 101
DNA aptamer HER2 protein DOX Breast cancer Yang et al. 2012 102
RNA aptamer EpCAM protein DOX Retinoblastoma Krishnakumar et al. 2012 103
RNA aptamer EGFR protein GEM Pancreatic cancer White et al. 2012 104

ALL: acute lymphoblastic leukemia; CCRF-CEM, T-acute lymphoblastic leukemia cell line; GEM, gemcitabine; LH86, human hepatocellular carcinoma cell line.