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. 2014 Mar 10;37(5):421–434. doi: 10.1111/jvp.12117

Table 2.

Pharmacokinetic parameters of imepitoin dosed to six beagle dogs at ascending doses of 10–100 mg/kg

Dose [mg/kg] Cmax [ng/mL] Tmax [h] AUCzero [ng·h/mL] Tlag obs [h]
10 1815 ± 920 8.67 ± 3.1 14 035 ± 8566 3.67 ± 0.92
20 3502 ± 1073 10.7 ± 4.0 33 551 ± 15 410 5.67 ± 0.95
50 6407 ± 1752 18.0 ± 3.8 73 081 ± 21 441 4.17 ± 1.05
100 13 554 ± 3333 8.67 ± 3.1 154 269 ± 49 882 2.25 ± 0.94

Pharmacokinetic parameters of imepitoin dosed to six beagle dogs (three male and three female dogs) single dose as micronized powder filled in enteric-coated gelatin capsules in an ascending dose design with at least 14 days washout between doses. Displayed is mean ± SEM of six animals.