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. 2014 Nov 24;172(1):1–23. doi: 10.1111/bph.12906
TARGETS
GPCRsa Enzymesb Transportersc
5-HT receptors adenylyl cyclases DAT
Adenosine A1 receptor Akt Catalytic receptorsd
Adenosine A2A receptor calpain ErbB (epidermal growth factor) receptor family
α1B-Adrenoceptor CaMKII ErbB-1
β1-Adrenoceptor CDK5 IGFR1
Dopamine D1 receptor ERK PDGFRβ
Dopamine D2 receptor Epac1 RTKs
Dopamine D3 receptor Epac2 TrkB
Dopamine D4 receptor GRK2 Ion channelse
Dopamine D5 receptor GSK3 GIRKs
Ghrelin receptor GSK3α Kir2 channels
Muscarinic M4 receptor GSK3β IP3 receptor
TA1 receptor MAPK Ligand-gated ion channelsf
PDK1 GluA1
PKA GluN2B
PKC Ionotropic glutamate receptors
PLC
PLCβ