| TARGETS | ||
|---|---|---|
| GPCRsa | Enzymesb | Transportersc |
| 5-HT receptors | adenylyl cyclases | DAT |
| Adenosine A1 receptor | Akt | Catalytic receptorsd |
| Adenosine A2A receptor | calpain | ErbB (epidermal growth factor) receptor family |
| α1B-Adrenoceptor | CaMKII | ErbB-1 |
| β1-Adrenoceptor | CDK5 | IGFR1 |
| Dopamine D1 receptor | ERK | PDGFRβ |
| Dopamine D2 receptor | Epac1 | RTKs |
| Dopamine D3 receptor | Epac2 | TrkB |
| Dopamine D4 receptor | GRK2 | Ion channelse |
| Dopamine D5 receptor | GSK3 | GIRKs |
| Ghrelin receptor | GSK3α | Kir2 channels |
| Muscarinic M4 receptor | GSK3β | IP3 receptor |
| TA1 receptor | MAPK | Ligand-gated ion channelsf |
| PDK1 | GluA1 | |
| PKA | GluN2B | |
| PKC | Ionotropic glutamate receptors | |
| PLC | ||
| PLCβ | ||