TARGETS | ||
---|---|---|
GPCRsa | Enzymesb | Transportersc |
5-HT receptors | adenylyl cyclases | DAT |
Adenosine A1 receptor | Akt | Catalytic receptorsd |
Adenosine A2A receptor | calpain | ErbB (epidermal growth factor) receptor family |
α1B-Adrenoceptor | CaMKII | ErbB-1 |
β1-Adrenoceptor | CDK5 | IGFR1 |
Dopamine D1 receptor | ERK | PDGFRβ |
Dopamine D2 receptor | Epac1 | RTKs |
Dopamine D3 receptor | Epac2 | TrkB |
Dopamine D4 receptor | GRK2 | Ion channelse |
Dopamine D5 receptor | GSK3 | GIRKs |
Ghrelin receptor | GSK3α | Kir2 channels |
Muscarinic M4 receptor | GSK3β | IP3 receptor |
TA1 receptor | MAPK | Ligand-gated ion channelsf |
PDK1 | GluA1 | |
PKA | GluN2B | |
PKC | Ionotropic glutamate receptors | |
PLC | ||
PLCβ |