Table 2.
Affinity of binding (pKi) of MOPr antagonists to MOPr expressed in HEK293 cells
| pKi | |
|---|---|
| GSK1521498 | 9.38 ± 0.10 (n = 7) |
| Naltrexone | 9.15 ± 0.04 (n = 6) |
| 6β-Naltrexol | 9.12 ± 0.09 (n = 6) |
Data are presented as mean ± SEM
Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.