Table 1. Properties of NFAT inhibitors.

Code	ChemB*	Nc3†	ID-Phos‡	GCR§	CN¶	IC50∥
1	114006	C	Phos.	C/N	Neg.	<25
2	115555	C	Phos	N	Neg.	10
3	115805	C	Phos	N	Neg.	<40
4	143072	C	Phos	N	Neg.	<25
5	149521	C	Phos	N	Neg.	<40
6	190027	C	De-Phos	N	Neg.	<10
7	202034	C	Phos	N	Neg.	14
8	205327	C	De-phos	N	Neg.	40
9	211950	C	Phos	N	Neg.	<20
10	219735	C	Phos	N	Neg.	15
11	228195	C	De-phos	N	Neg.	22
12	232755	C	De-phos	N	Neg.	32
13	156381	C	Phos	N	Neg.	15
14	103885	C	Phos	N	Neg.	<10

^*Chembridge Corporation code for compounds.

^†Effect on NFATc3 localization in the presence of calcium ionophore (C, cytoplasmic, N, nuclear).

^‡Effect on NFATc3 phosphorylation status in the presence of ionomycin.

^§Effect on the dexamethasone-induced translocation of the glucocorticoid receptor to the nucleus (C, cytoplasmic; N, nuclear).

^¶Effect on calcineurin in vivo. Neg., negative.

^∥Apparent concentration of inhibitor at which 50% of NFATc3 fails to enter the nucleus.