Skip to main content
. 2014 Mar 24;16(6):560–568. doi: 10.1111/dom.12281

Table 2.

Concomitant therapies at screening

% Normal renal function* Mild RI* Moderate RI*
Linagliptin 5 mg (n = 870) Placebo (n = 342) Linagliptin 5 mg (n = 620) Placebo (n = 218) Linagliptin 5 mg (n = 68) Placebo (n = 25)
Subjects with ≥1 specific drug 66.7 70.5 81.0 80.7 88.2 88.0
ASA 30.5 34.2 37.6 38.1 29.4 48.0
Antihypertensives 51.1 52.6 69.5 70.2 82.4 84.0
 β-blockers 14.9 16.4 23.9 26.1 30.9 20.0
 ACE inhibitors 26.9 26.9 30.0 31.7 33.8 48.0
 Diuretics 8.7 9.6 18.5 14.7 32.4 32.0
 ARBs 10.5 10.8 16.6 13.3 19.1 16.0
 Calcium antagonists 11.0 11.7 20.2 19.7 27.9 24.0
 Combinations 5.9 7.3 12.9 12.4 17.6 24.0
Lipid-lowering drugs 34.5 38.3 43.7 41.7 51.5 40.0
 Niacin 1.6 0.3 1.1 0.5 0 0
 Fibrates 4.8 7.0 7.6 7.3 7.4 16.0
 Statins 30.0 31.9 37.4 35.8 45.6 32.0
 Other 2.3 2.6 2.6 0.5 1.5 4.0
Glucose-lowering drugs
 Treatment-naïve 8.3 11.4 15.6 22.9 10.3 4.0
 Metformin only 28.3 27.5 29.0 30.3 25.0 24.0
 SU only 1.8 3.2 3.1 2.3 1.5 8.0
 Metformin + SU 59.8 56.4 50.6 43.1 60.3 64.0
 Others 1.8 1.5 1.6 1.4 2.9 0

ACE, angiotensin-converting enzyme; ARBs, angiotensin receptor blockers; ASA, acetyl salicylic acid; MDRD, modification of diet in renal disease; RI, renal impairment; SU, sulphonylurea.

Renal function according to MDRD formula: normal, ≥90 ml/min/1.73 m2; mild, 60–<90 ml/min/1.73 m2; moderate, 30–<60 ml/min/1.73 m2.

Including mono- and combination therapies.