TABLE 1.
Parameter | MIC or MBC (μM) |
||
---|---|---|---|
TBA-354 | Pa | Delamanid | |
MIC (replicating) | 0.006 | 0.04 | 0.002 |
MBC (replicating) | 0.006 | 0.061 | 0.003 |
LORA (NR) MICa | 0.27 | 2.28 | 0.7 |
LORA (NR) MBC | 3.4 | 17.4 | 4.4 |
4% BSAb MIC (replicating) | 0.011 | 0.072 | 0.006 |
10% FBSc MIC (replicating) | 0.012 | 0.038 | 0.009 |
Clofazimine, 1.42 μM; thioridazine, 11.74 μM; capreomycin, 5.92 μM, linezolid, 28.42 μM; INH and ethambutol, >1,000 μM.
BSA, bovine serum albumin.
FBS, fetal bovine serum.