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. 2014 Nov 26;12(1):46–55. doi: 10.1021/mp500405h

Figure 1.

Figure 1

Inhibitors of GLS1 and TG2. 968 and BPTES are reversible allosteric regulators of GLS1. MDC is a reversible inhibitor of TG2, which serves as an amine-bearing substrate. T101 and Z-Don are irreversible inhibitors of TG2, which bind at the catalytic site. All inhibitors are cell permeable except for T101.