Table 1.
Average Number of CDs per PRTx, Threading Efficiencies, Yields, and Free CD Content
β-CD PRTx | base MW (Da) | PEG:PPG | # CDs | % threading | % yield | % free CD |
---|---|---|---|---|---|---|
F127 | 12,500 | 200:65 | 15 | 71.4 | 32.9 | 4.4 |
F68 | 8,350 | 151:29 | 14 | 100 | 13.3 | 3.6 |
L64 | 2,900 | 26:30 | 12 | 92 | 29.1 | 2.4 |
L35 | 1,900 | 22:16 | 5 | 63 | 19.1 | 1.2 |