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. 2014 Dec 5;58(1):466–479. doi: 10.1021/jm501603h

Table 2. Summary of the Number of Small Molecule Inhibitors of Each Type Bound to Classical DFG-Out Conformations.

inhibitor class total number of inhibitor bound classical DFG-out conformations number of unique inhibitors
type I 47 42
type II 185 147
type III 2 2