Figure 1. Schematic representation of the Akt kinase reporter (BAR).
A, The chimeric Akt kinase reporter is a fusion of the N-Luc and C-Luc luciferase protein linked to an Akt peptide domain containing the Akt substrate sequence and a yeast FHA2 phospho-Ser/Thr binding domain. B, Phosphorylation of the Akt substrate peptide in the reporter results in interaction with the FHA2 phospho-peptide binding domain leading to steric constraints on the N-Luc and C-Luc. Inhibition of Akt kinase activity results in decreased binding of phospho-peptide and the binding domain which enables reconstitution of luciferase and restored bioluminescence.
