| 2000 Linezolid | 2004 Gemifloxacin | 2009 Tebipenem pivoxil |
| 2001 Telithromycin | 2005 Doripenem | 2009 Telavancin |
| 2002 Biapenem | 2005 Tigecycline | 2009 Antofloxacin |
| 2002 Ertapenem | 2007 Retapamulin | 2009 Besifloxacine |
| 2002 Prulifloxacin | 2007 Garenoxacin | 2010 Ceftaroline fosamil |
| 2002 Pazufloxacin | 2008 Ceftobiprole medocaril | 2011 Fidaxomicin |
| 2002 Balofloxacin | 2008 Sitafloxacin | 2012 Bedaquiline |
| 2003 Daptomycin |