Table 3.
Effect of ML-7 and Cytochalasin D on Nav1.5 parameters
| ML-7 | Cytochalasin D | |||
|---|---|---|---|---|
| WT (n=15) | D117N (n=10) | WT (n=10) | D117N (n=11) | |
| Peak current density (pA/pF) | -231.6 [-288.4; -193.9] | -230.8 [-282.3; -159.1] | -143.8 [-219.6; -120.2] | -203.0 [-234.0; -177.3] | 
| Activation | ||||
| Vh (mV) | -36.2 [-38.7; -35.2] | -42.2 [-47.2; -39.4] | -34.8 [-35.3; -26.9] | -45.7 [-50.2; -36.2] | 
| k | 7.5 [5.7; 8.3] | 7.4 [6.8; 7.8] | 8.3 [7.1; 10.4] | 6.7 [6.5; 7.4] | 
| Fast-inactivation | ||||
| Vh (mV) | -99.9 [-104.6; -96.4] | -95.0 [-101.7; -91.2] | -93.9 [-103.0; -88.8] | -97.9 [-106.0; -95.1] | 
| k | 6.8 [6.3; 7.2] | 6.2 [5.6; 7.1] | 7.1 [5.4; 7.7] | 5.8 [5.6; 6.6] | 
Vh, represents midpoint voltage of maximal activation/inactivation; k, slope factor; n, the number of patches.