Table 1.
Receptor | n | pEC50 ± SEM | Emax ± SEM | pIC50 ± SEM | Selectivity |
---|---|---|---|---|---|
α7 | 18 | 7.41 ± 0.09 | 73 ± 4.1% | ||
α1β1γδ | 6 | 4.97 ± 0.05 | 274 | ||
α4β2 | 6 | 5.40 ± 0.07 | 101 | ||
α3β4 | 5 | 5.28 ± 0.08 | 144 | ||
5-HT3 | 6 | 4.72 ± 0.09 | 488 |
Receptor | n | pEC50 ± SEM | Emax ± SEM | pIC50 ± SEM | Selectivity |
---|---|---|---|---|---|
α7 | 18 | 7.41 ± 0.09 | 73 ± 4.1% | ||
α1β1γδ | 6 | 4.97 ± 0.05 | 274 | ||
α4β2 | 6 | 5.40 ± 0.07 | 101 | ||
α3β4 | 5 | 5.28 ± 0.08 | 144 | ||
5-HT3 | 6 | 4.72 ± 0.09 | 488 |