Table XIV.
Cytotoxicity Data for Arylamino Analogs 431–446
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---|---|---|---|---|
IC50 (μM) |
||||
Compound | Colo 205 | Hop62 | HT1080 | DWD |
PPT | 5.0 | 13.1 | 8.1 | 6.1 |
431 | 8.1 | >80 | 8.2 | 22 |
432 | 2.7 | 30.1 | 9.7 | 2.3 |
434 | 8.3 | 8.6 | >80 | 6.5 |
437 | 7.0 | 15.2 | 9.5 | 5.2 |
441 | 7.1 | 60.3 | 9.1 | 7.3 |
442 | 8.3 | 10.1 | >80 | 9.1 |