Table XXI.
Cytotoxicity Data for Indole-Substituted Analogs 568–574
| |||||
|---|---|---|---|---|---|
| IC50 (μM) |
|||||
| Compound | HeLa | K562 | K562/AO2 | KB | KBV |
| ETO | 2.11 ± 1.17 | 0.9 ± 0.08 | 7.05 ± 5.08 | 3.36 ± 1.05 | 55.47 ± 4.36 |
| 568 | 1.05 | 0.99 ± 0.60 | 4.04 ± 0.97 | 3.99 ± 1.28 | 6.28 ± 2.05 |
| 569 | 5.237 | 0.29 ± 0.19 | 0.12 ± 00.6 | 2.49 ± 0.94 | 3.49 ± 1.05 |
| 570 | 3.805 | 0.23 ± 0.16 | 0.70 ± 0.02 | 0.88 ± 0.23 | 3.62 ± 2.17 |
| 571 | 0.15 | 0.40 ± 0.14 | 0.29 ± 0.26 | 1.00 ± 0.78 | 3.16 ± 1.46 |
| 572 | 0.73 | 1.22 ± 0.35 | 0.62 ± 0.28 | 4.99 ± 1.36 | 5.46 ± 3.65 |
| 573 | 10.67 | 0.31 ± 0.18 | 0.22 ± 0.20 | 1.03 ± 0.38 | 2.59 ± 0.28 |
| 574 | 11.11 | 0.46 ± 0.37 | 0.10 ± 0.01 | 1.62 ± 1.25 | 2.30 ± 2.17 |
Cytotoxicity against HeLa, KB, and KBV cell lines and against K562 and K562/AO2 cell lines measured by standard MTT and SRB assay methods, respectively.
Each value represents mean ± SD of three independent experiments.