Skip to main content
. Author manuscript; available in PMC: 2016 Jan 1.
Published in final edited form as: Med Res Rev. 2014 May 14;35(1):1–62. doi: 10.1002/med.21319

Table XXVII.

Cytotoxicity Data for Triazole Analogs 674–682

graphic file with name nihms-662637-t0054.jpg
IC50 (μM)
Compound DU-145 PC-3 A549 HCT-15 HOP-62 SF-295
ETO 2.97 100 7.63 1 4.8 5.69
674 25.8 127 125 15 NTa 26.8
675 42 221 556 NT 142 35.1
676 237 316 59.9 16 178 14.5
677 18.6 94.9 51.8 237 121 53.4
678 26.5 268 114 NT NT 88
679 3.11 34.6 3 0.93 8.55 2.01
680 4.95 24.3 6.88 1 5.27 16.1
681 2.73 8.62 7.33 3.57 5.96 2.51
682 5.04 20.8 7.04 2.14 16.2 8.29
a

NT, not tested.