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. 2014 Dec 18;20(2):87–98. doi: 10.1016/j.rpor.2014.11.010

Table 2.

Silk-based drug delivery systems for cancer therapy.

Silk biomaterial Preparatiom method Drug/route of administration Target Cell line/in vivo model References
B. mori silk film Film casting with water vapor annealing Doxorubicin/intratumoral Breast cancer MDA-MB-231/orthotopic adrenal tumor xenograft in mice 15,24
B. mori silk hydrogel Self-assembly mediated by sonication Doxorubicin/intratumoral Breast cancer MDA-MB-231, MCF-7/tumor xenograft in mice 16
B. mori silk particle Self-assembly with paclitaxel solution in ethanol Paclitaxel/intratumoral Gastric cancer BCG-823/tumor xenograft in mice 20
B. mori silk particle Desolvation method with acetone Doxorubicin Breast cancer MCF-7/n/a 18
B. mori silk-albumin particle Desolvation with acetone and crosslinking with glutaraldehyde Metotrexate Breast cancer MDA-MB-231/n/a 21
B. mori silk fibroin particle and silk fibroin-chitosan particles The microdot capillary method, lyophilization, methanol treatment Curcumin Breast cancer, melanoma MCF-7, MDA-MB-453/n/a 22
B. mori silk film coated liposome Lyophilization of silk fibroin with emodin-loaded liposomes and methanol treatment Emodin Breast cancer, melanoma MCF-7, MDA-MB-453, BT-474/n/a 17,30
Bioengineered silk fibroin–elastin-like particle Self-assembly with hydrophobic doxorubicin Doxorubicin Cervical cancer HeLa/n/a 34
Bioengineered functionalized spider silk sphere Salting-out with potassium phosphate Doxorubicin Her2/neu overexpressing ovarian and breast cancer SKOV3, SKBR3/n/a 40
Bioengineered spider silk and DNA complexes Self- assembly with DNA Plasmid DNA/intravenous Breast cancer, melanoma MDA-MB-231, MDA-MB-435/tumor xenograft in mice 38,39