ATL-801 (78) |
A2B antagonist |
DSS colitis, IL-10 KO spontaneous colitis |
Kolachala V et al, 2008 96 (ameliorates colitis) |
PSB-1115 (27) |
A2B antagonist |
DSS colitis |
Frick JS et al, 2009 68 (exacerbates colitis) |
IB-MECA (9) |
A3 agonist |
IL-10 KO, DSS colitis |
Gessi S et al, 2008 242
|
ATL-146e (69) |
A2A agonist |
Rabbit colitis, spont. Ileitis in SAMP1/YitFc mice |
Odashima M et al, 2005132
|
4-amino-2-(2-hydroxyl-1-decyl) pyrazole[3,4-d]pyrimidine (APP) (63) |
AdoDase inhibitor |
DNBS-induced colitis |
Antonioli L et al, 2007 49
|
Pentostatin (62) |
AdoDase inhibitor |
Severe IL-10−/− colitis with piroxicam-induced colitis |
Brown JB et al, 2008 243
|
Dipyridamole (61) |
ENT1, ENT2 inhibitor |
LPS/phytohaemagglutinin-induced gut mononuclear cells from CD patients |
Poturoglu S et al, 2009 83
|
MRS2500 (51) |
P2Y1 antagonist |
Neurogenic secretion model (in vitro) |
Fang X et al, 2006 103
|