Skip to main content
. Author manuscript; available in PMC: 2015 Mar 13.
Published in final edited form as: J Med Chem. 2011 Dec 7;55(1):437–448. doi: 10.1021/jm2013198

Scheme 3. a.

Scheme 3. a

aReaction conditions: (a) CDI (5 equiv), DMF, room temp 3 h; (b) dry MeOH (5 equiv), room temp 8 min; (c) NDP(α-B), MgCl2 (8 equiv), room temp overnight.