. Author manuscript; available in PMC: 2015 Mar 20.

Published in final edited form as: Curr Med Chem. 2012;19(24):4194–4206. doi: 10.2174/092986712802430036

Table 2.

PRCP Inhibition Data (N-Substituted-Pro-Pro-NH dodecylamides)


Cpnd	R	rPRCP K_i (µM)	PRCP-Dependent PK Activation on HPAEC K_i (µM)
3(UM8190)	H	43.08 ± 3.6	34.07 ± 4.3
4a		NE	NE
4b		NE	NE
4c		NE	NE
4d		NE	NE
4e		NE	NE