Table 1. List of the available ligands co-crystallized with ALK receptor.
Molecular Structure | Ligand name | PDB ID (resolution) | Reference |
---|---|---|---|
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Piperidine-carboxamide | 4DCE (2.03Å) | (27) |
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Piperidine-carboxamide | 4FNZ (2.60Å) | (26) |
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PHA-E429 | 2XBA (1.95Å) | (22) |
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NVP-TAE684 | 2XB7 (2.50Å) | (22) |
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Acyliminobenzimidazole inhibitor 36 | 4FOD (2.00Å) | (28) |
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Acyliminobenzimidazole inhibitor 1 | 4FOB (1.90Å) | (28) |
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Acyliminobenzimidazole inhibitor 2 | 4FOC (1.70Å) | (28) |
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Crizotinib | 2XP2(1.90Å) | (29) |
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CH5424802 | 3AOX(1.75Å) | (30) |