Skip to main content
. 2015 Jan 29;4(2):494–507. doi: 10.1039/c4tx00160e

Table 3. Specific inhibitors used in efflux transporter inhibition studies.

Efflux transporter Inhibitor Concentration range (μM) Solvent (maximum concentration)
MDR1 Cyclosporine A 0.01–20 DMSO (0.1%)
MRP2 Probenecid 0.5–1000 NaOH (0.01%)
BCRP Sodium taurocholate 1–1500 Sterile dH2O
BSEP Ko 143 0.01–20 DMSO (0.4%)