Skip to main content
. Author manuscript; available in PMC: 2016 Jan 31.
Published in final edited form as: JACC Cardiovasc Imaging. 2015 Feb;8(2):210–220. doi: 10.1016/j.jcmg.2014.12.008

Table 2.

Studies Not Meeting Inclusion Criteria but with Assessments of Microvascular Function

Treatment Baseline CFR <2.5 No CAD ≥50% stenosis Mode of Assessing CFR or MPR Patients (n) Findings Authors
Renin/Angiotensin/Aldosterone Inhibitors
Eplerenone 25 mg No Yes IC Doppler 25 Angina ↔, CFR ↔ Bavry et al. 2014 (44)
Candesartan 4–8mg NA No IC Doppler 14 CFR ↑ Iino et al. 2012 (74)
Enalapril 5mg 2x daily No Yes IC Doppler 10 Angina ↑, CFR ↑ Chen et al. 2002 (75)
Enalapril 10mg–20mg/day No Yes Argon Dilution 15 Symptoms ↑, CFR ↑ Motz et al. 1996 (43)
Enalapril 5mg 2x daily No Yes PET 10 Exercise capacity ↑ Kaski et al. 1994 (42)
Statins
Fluvastatin 40mg Yes Yes TTDE 23 Angina ↑, CFR ↑ Zhang et al. 2014 (50)
Atorvastatin 80mg No No IC Doppler 20 CFR ↔ Eshtehardi et al. 2012 (52)
Atorvastatin 20mg Yes Yes TTDE 20 CFR ↑ Caliskan et al. 2007 (51)
Nitric Oxide Modulators
L-Arginine infusion 1 time infusion No Yes IC Doppler 11 CBF ↓ Gellman et al. 2004 (58)
Tetrahydrobiopterin 1 time infusion No No IC Doppler 23 CBF ↑ Setoguchi et al. 2001 (76)
L-Arginine infusion 3gm 3x daily No No IC Doppler 13 Angina ↑, CFR ↔ Lerman et al. 1998 (59)
L-Arginine infusion 1 time infusion No No IC Doppler 8 CBF ↑ Egashira et al. 1996 (57)
Calcium Blockers
Diltiazem 90mg No Yes TTDE 23 Angina ↑, CFR ↑ Zhang et al. 2014 (50)
Lidoflazine 240 to 360mg No Yes Thermodilution 11 Angina ↔, MBF ↑, Arrhythmias* Cannon et al. 1990 (48)
Verapamil 80mg 4x daily No Yes Thermodilution 17 Angina ↑ Cannon et al. 1985 (47)
Nifedipine 10mg 4x daily No Yes Thermodilution 9 Angina ↑ Cannon et al. 1985 (47)
Alpha blockers
Doxazosin 2mg No Yes PET Scan 11 Angina ↔, CBF ↔, Rosen et al. 1999 (61)
Anti-Anginals & Nitrates
Ivabradine 5mg Yes Yes TTDE 16 Angina ↑, CFR ↔ Villano et al. 2013 (68)
Isosorbide dinitrate 5mg (SL) NA Yes TTDE 29 Stress Testing ↔ Russo et al. 2013 (69)
Ranolazine 500 mg – 1000mg No Yes CMR 20 Angina ↑, CFR ↔ Mehta et al. 2011 (67)
Isosorbide dinitrate 10mg (SL), 2mg (IV) NA Yes Thermodilution 11 Angina ↓, CBF ↓ Bugiardini et al. 1993 (70)
Estrogens
17β-estradiol 1mg + drospirenone 2mg No NA PET 27 MPR ↑ Knuuti et al. 2007 (63)
Devices
EECP Yes Yes TTDE 24 Angina ↑, CFR ↑ Luo et al. 2012 (65)
TENS NA Yes IC Doppler 13 CBF ↓ Sanderson et al. 1996 (66)
Other
Bariatric Surgery Yes NA TTDE 50 CBF ↑ Nerla et al. 2012 (71)
Congac No NA TTDE 18 CFR ↔ Kiviniemi et al. 2008 (77)
Vitamin C 3g infusion No NA PET 19 CFR ↑ in asymptomatic smokers Kaufmann et al. 2000 (78)
Exercise Training No No PET 13 CFR ↑ Czernin et al. 1995 (79)

Studies of therapies in patients who did not meet strict inclusion criteria nor had evidence of structural heart disease, heart failure, or untreated HTN, but which did assess coronary microvascular function.

TTDE = transthoracic Doppler echocardiography, IC = intracoronary, PET = positron emission tomography, CFR = coronary flow reserve, MPR = myocardial perfusion reserve, CBR = coronary blood flow, EECP = enhanced external counterpulsation, SL = sublingual, IV = intravenous

(↑) = improved with therapy; (↔) = not statistically different; (↓) = worse with therapy (NA) = not assessed

(*) = treatment intervention associated with increased risk of arrhythmias.