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. Author manuscript; available in PMC: 2016 Apr 15.
Published in final edited form as: Bioorg Med Chem Lett. 2015 Mar 2;25(8):1761–1764. doi: 10.1016/j.bmcl.2015.02.055

Table 2.

Validation of radioiodinated drugs by radioligand saturation studies using mouse brain homogenates.

compound yielda KD (nM) literature KD
(nM)
[125I]IPAG 29 10.3 ± 4.4 8.7 – 11.21h
[125I]4-I-Clonidine 11 0.11 ± 0.03 0.46 ± 0.0612b
[125I]AM251 33 0.46 ± 0.01 0.23 – 0.6212a
a

average radiochemical yield based on two repetitions.