Table 2.
compound | yielda | KD (nM) | literature KD (nM) |
---|---|---|---|
[125I]IPAG | 29 | 10.3 ± 4.4 | 8.7 – 11.21h |
[125I]4-I-Clonidine | 11 | 0.11 ± 0.03 | 0.46 ± 0.0612b |
[125I]AM251 | 33 | 0.46 ± 0.01 | 0.23 – 0.6212a |
average radiochemical yield based on two repetitions.