Table 3.
C–C Activation of 2-Cyclopropylpyridines with Pd(OAc)2/PhI(OAc)2
| ||
|---|---|---|
|
| ||
| entry | R | Yield |
| 1 | 4-CH3 (6) | nd |
| 2 | 6-CH3 (7) | nd |
| 3 | 3-CH3 (8) | 29% |
| 4 | 3-CH3CH2 (9) | 21% |
| 5 | 3-CH3O (10) | 34% |
C–C Activation of 2-Cyclopropylpyridines with Pd(OAc)2/PhI(OAc)2
| ||
|---|---|---|
|
| ||
| entry | R | Yield |
| 1 | 4-CH3 (6) | nd |
| 2 | 6-CH3 (7) | nd |
| 3 | 3-CH3 (8) | 29% |
| 4 | 3-CH3CH2 (9) | 21% |
| 5 | 3-CH3O (10) | 34% |