Table 1.
nAChR subtype | Ki, nM | α7-nAChR Binding selectivity |
---|---|---|
α7 (rat) | 0.5 ± 0.2 | |
α3β4 (human) | 45 ± 8 | α7/α3β4 = 90 |
α4β2 (human) | 1707 ± 373 | α7/α4β2 = 3,414 |
nAChR subtype | Ki, nM | α7-nAChR Binding selectivity |
---|---|---|
α7 (rat) | 0.5 ± 0.2 | |
α3β4 (human) | 45 ± 8 | α7/α3β4 = 90 |
α4β2 (human) | 1707 ± 373 | α7/α4β2 = 3,414 |