Table 2.
Kinetic constants for 4, 8, 9, and 11
l-NIO (4) | 8 | 9 | 11 | |
---|---|---|---|---|
kinact(min−1) | 0.073 ± 0.003 | 0.0743 ± 0.0073 | 0.131 ± 0.0095 | 0.347 ± 0.006 |
KI(μM) | 13.7 ± 1.6 | 243 ± 31.4 | 674 ± 80 | 4009 ± 426 |
kinact/KI
(μM−1.min−1) |
0.0053 ± 0.0007 | 0.00031 ± 0.000028 | 0.00020 ± 0.0000096 | 0.000087 ± 0.000011 |