Table 1.
Chemical structures and IC50 values of AI-10-49 and related compounds, determined by using the FRET assay.
Compound Name | Compound Structure | FRET IC50 (μM) |
---|---|---|
AI-4-88 |
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>240 |
AI-4-57 |
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22 ± 8 |
AI-10-11 |
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14 ± 4 |
AI-10-19 |
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>2.5 |
AI-4-83 |
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0.35 ± 0.05 |
AI-4-82 |
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0.44 ± 0.07 |
AI-4-71 |
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0.37 ± 0.07 |
AI-10-47 |
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2.0 ± 0.03 |
AI-10-49 |
![]() |
0.26 ± 0.01 |