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. Author manuscript; available in PMC: 2016 May 20.
Published in final edited form as: Tetrahedron Lett. 2015 May 20;56(21):2832–2835. doi: 10.1016/j.tetlet.2015.04.061

Table 2.

Pyrazololo analogs tested against TbrPDEB1

graphic file with name nihms685683t11.jpg
Cpd R R1 TbrPDEB1 (% inh)a
18a graphic file with name nihms685683t12.jpg H 0
18b graphic file with name nihms685683t13.jpg graphic file with name nihms685683t14.jpg 5 ± 3
a

Data shown are average of 2 replicate independent experiments. Compounds were tested at 10 µM concentrations.