Table 3.

Scope of aryl iodide reagents for the enantioselective arylation of cyclopropylmethylamines^a,^b

^aExperiments were performed with 1 (0.2 mmol), aryl iodide (0.6 mmol), Pd(OAc)₂ (0.02 mmol), Ag₂CO₃ (0.4 mmol), sodium trifluoroacetate (0.1 mmol), Boc-L-Val-OH (0.04 mmol) in t-BuOH (1 mL) for 18 hours at 80 ºC under air.

^bIsolated yields.