Table 3.
Percentages of ionizable residues in receptor proteins that exhibit substantial pK change (|ΔpK | > 1) upon ligand binding in the biologically relevant pH range from 4 to 8. Adopted from Aguilar et al.1
Complex type | Minimum | Average | Maximum |
---|---|---|---|
Protein-protein (20) | 1.5% | 8.7% | 16.7% |
Protein-small molecule (20) | 2.1% | 5.7% | 12.5% |
Protein-nucleic acid (20) | 5.6% | 12.3% | 24.4% |