Table 4.
Entry | Aryne | Geometry-optimized structurea | Site of attack (angle difference) |
---|---|---|---|
1 | C5 (4°) | ||
2 | C4 (10°) | ||
3 | C4 (13°) | ||
4 | C4 (7°) | ||
5 | C4 (6°) | ||
6 | N/A (0°) |
Geometry optimizations were performed using DFT methods (B3LYP/6-31G*; B3LYP/LACVP was used for 6-iodo-4,5-indolyne (entry 6)).