. Author manuscript; available in PMC: 2016 Feb 4.

Published in final edited form as: J Am Chem Soc. 2015 Jan 15;137(4):1408–1411. doi: 10.1021/ja512306a

Table 3. Substrate scope with different amines^a.

All yields are isolated yields.

4% of ortho-C–H vinylation product and 3% of sequential C–H/C–C activation product were observed.

6% of ortho-C–H vinylation product was observed.

2.0 equiv of alkyne 2a was used.

The reaction conversion was 83%, determined by crude ¹H NMR.

Table 3. Substrate scope with different aminesa.