Table 4.
IC50 in IU/ml
| Cell line | dm HpA | wt HpA | L-ASP | ERWase |
|---|---|---|---|---|
| SupB15 | 0.0043 | 0.0033 | 0.0032 | 0.0030 |
| RS4;11 | 0.0055 | 0.0052 | 0.0054 | 0.0057 |
| MOLT-4 | 0.0108 | 0.0097 | 0.0088 | 0.0039 |
| SEM | nd | 2.05 | 1.14 | 0.07 |
| BV173 | nd | 5.21* | 4.72* | 0.34 |
| HL-60 | nd | 5.39* | 4.62* | 0.51 |
| SD-1 | nd | nd | 10.54* | 0.55 |
| REH | nd | 5.26* | 3.13 | 0.35 |
| RCH-ACV | nd | 6.67* | 11.82* | 1.13 |
| NALM6 | nd | 12.62* | 10.56* | 1.40 |
| K-562 | nd | nd | nd | 5.37* |
IC50s were calculated from normalized data (Fig 2) using non-linear regression with GraphPad Prism.
extrapolated for values > 3 IU/ml, n=4–5 for each cell line, nd: not determined >100 IU/ml.