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. Author manuscript; available in PMC: 2015 Jun 15.
Published in final edited form as: Nanomedicine. 2012 Jun 6;9(1):1–14. doi: 10.1016/j.nano.2012.05.013
Application(s)/Product(s) Company Status Condition Nanocomponent Targeting Mechanism
Ontak [45,46] Seragen, Inc. Approved (1999) T-Cell Lymphoma Protein Nanoparticle IL-2 Protein
MBP-Y003, MBP-Y004, MBP-Y005 [47] Mebiopharm Co., Ltd Preclinical Lymphoma Liposome Transferrin
MBP-426 [4749] Mebiopharm Co., Ltd Phase I/II Solid Tumors Liposome Transferrin
CALAA-01 [19,50] Calando Pharmaceuticals Phase I Solid Tumors Nanoparticle Transferrin
SGT-53 [19,51] SynerGene Therapeutics, Inc. Phase I Solid Tumors Liposome Transferrin
MCC-465 [48,52] Mitsubishi Tanabe Pharma Corp Phase I Stomach Cancer Liposome GAH Antibody
Actinium-225-HuM195 [53] National Cancer Institute Phase I Leukemia Nanoparticle HuM195 Antibody
AS15 [54] GlaxoSmithKline Biologicals Phase I/II Metastatic Breast Cancer Liposome dHER2 Antibody
PK2 [48,55] Pharmacia & Upjohn Inc. Phase I Liver Cancer Polymeric Nanoparticle Galactose
Rexin-G, Reximmune-C [56,57] Epeius Biotechnologies Phase I/II Solid Tumors Nanoparticle von Willebrand factor (Collagen-Binding)
Aurimune (CYT-6091) [19,58]
Auritol (CYT-21001) [59]
CytImmune Sciences, Inc. Phase II Preclinical Solid Tumors Colloid Gold TNF-α
SapC-DOPS[60,61] Bexion Pharmaceuticals, Inc. Preclinical Solid Tumors Liposome Saposin C
Targeted Emulsions [62,63] Kereos, Inc. Preclinical In Vivo Imaging Emulsion "Ligands"

Opaxio [42,64] Cell Therapeutics, Inc. Phase III Solid Tumors Polymeric Nanoparticle Enzyme-Activated
ThermoDox [43] Celsion Corporation Phase II/III Solid Tumors Liposome Thermosensitive
DM-CHOC-PEN [44,65] DEKK-TEC, Inc. Phase I Brain Neoplasms Emulsion Penetrate Blood-Brain-Barrier