Table 4.
Various analogs
| Cmp | Structure | IC50(μM)a |
|---|---|---|
| 3 |
|
>25 |
| 4 |
|
>25 |
| 5 |
|
>25 |
| 6 |
|
0.80 |
| 7 |
|
0.18 |
| 8 |
|
0.63 |
| 9 |
|
>25 |
| 10 |
|
>25 |
| 11 |
|
8.0 |
| 12 |
|
9.9 |
Average of at least two measurements in DiI uptake assay.
Various analogs
| Cmp | Structure | IC50(μM)a |
|---|---|---|
| 3 |
|
>25 |
| 4 |
|
>25 |
| 5 |
|
>25 |
| 6 |
|
0.80 |
| 7 |
|
0.18 |
| 8 |
|
0.63 |
| 9 |
|
>25 |
| 10 |
|
>25 |
| 11 |
|
8.0 |
| 12 |
|
9.9 |
Average of at least two measurements in DiI uptake assay.