Skip to main content
. Author manuscript; available in PMC: 2016 Jun 15.
Published in final edited form as: Bioorg Med Chem Lett. 2015 Apr 11;25(12):2594–2598. doi: 10.1016/j.bmcl.2015.03.074

Table 1.

Amide analogs

graphic file with name nihms689082u2.jpg
Cmp R1 IC50 (μM)a
1a graphic file with name nihms689082t1.jpg 0.055±0.014
1c graphic file with name nihms689082t2.jpg 0.81
1e graphic file with name nihms689082t3.jpg 17
1g graphic file with name nihms689082t4.jpg 7.1
1b graphic file with name nihms689082t5.jpg 0.20
1d graphic file with name nihms689082t6.jpg 0.42
1f graphic file with name nihms689082t7.jpg 1.6
a

Average of at least two measurements in DiI uptake assay, ± standard error of mean when n > 2.