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. Author manuscript; available in PMC: 2016 Jun 15.
Published in final edited form as: Bioorg Med Chem Lett. 2015 Apr 11;25(12):2594–2598. doi: 10.1016/j.bmcl.2015.03.074

Table 2.

Tetrazole replacements

graphic file with name nihms689082u3.jpg
Cmp Ar1 IC50 (μM)a
1a graphic file with name nihms689082t8.jpg 0.055±0.014
2b graphic file with name nihms689082t9.jpg 0.13
2d graphic file with name nihms689082t10.jpg 0.023
2a graphic file with name nihms689082t11.jpg 37
2c graphic file with name nihms689082t12.jpg 6.3
a

Average of at least two measurements in DiI uptake assay, ± standard error of mean when n > 2.