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. Author manuscript; available in PMC: 2016 Jun 15.
Published in final edited form as: Bioorg Med Chem Lett. 2015 Apr 11;25(12):2594–2598. doi: 10.1016/j.bmcl.2015.03.074

Table 3.

Arene SAR

graphic file with name nihms689082u4.jpg
Cmp Ar2 IC50 (μM)a
1a graphic file with name nihms689082t13.jpg 0.055±0.014
3b graphic file with name nihms689082t14.jpg 0.18
3d graphic file with name nihms689082t15.jpg >25
3f graphic file with name nihms689082t16.jpg 3.8
3h graphic file with name nihms689082t17.jpg 0.17
3j graphic file with name nihms689082t18.jpg 0.18
3l graphic file with name nihms689082t19.jpg 0.23
3a graphic file with name nihms689082t20.jpg 0.37
3c graphic file with name nihms689082t21.jpg 0.38
3e graphic file with name nihms689082t22.jpg 0.62
3g graphic file with name nihms689082t23.jpg 0.49
3i graphic file with name nihms689082t24.jpg 0.13
3k graphic file with name nihms689082t25.jpg 0.027±0.008
a

Average of at least two measurements in DiI uptake assay, ± standard error of mean when n > 2.