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. Author manuscript; available in PMC: 2015 Jul 2.
Published in final edited form as: J Am Chem Soc. 2015 Mar 9;137(10):3715. doi: 10.1021/jacs.5b00787
graphic file with name nihms674325u1.jpg

R dr

C6H5 (2a) 8–14:1
4-ClC6H4 (2b) 14:1
4-MeC6H4 (2c) 11:1
4-MeOC6H4 (2d) 10:1
4-NCC6H4 (2e) 17:1
2-MeC6H4 (2f) 6:1
benzo[d][1,3]dioxol-5-yl (2g) 20:1
fur-2-yl (2h) 6:1
N-Ts-indol-3-yl (2i) 25:1
N-Boc-indol-3-yl (2j) 20:1