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. 2014 Sep 4;53(42):11376–11380. doi: 10.1002/anie.201404921

Table 1.

Molar fractions of bound ligands for different ligand/protein ratios and experimentally observed contrast CLLS for a titration of vanillic acid diethylamide (ligand II, KD=790 μm) in the presence of the protein Hsp90.

[L]tot/[P]tot Xbound [mol %] Contrast CLLS [%]
56 0.74 72
125 0.49 63
202 0.36 54
272 0.28 45
366 0.22 41
548 0.16 29
707 0.13 23