Table 1. Summary of labeled versus unlabeled plate data.
NT, not tested; NI, not included.
Score of labeled/unlabeled | ||||||||
---|---|---|---|---|---|---|---|---|
ID | 4 | 5 | 6 | 7 | 89 | Unique leads | Leads tested | Testedcrystals |
Tt46: ssDNA-specific exonuclease | 31 | 13/6 | 1/1 | 1/0 | 0/0 | 22 | 22 | 7 |
Tt55: translation initiation factor | 31 | 26/21 | 12/14 | 3/1 | 3/3 | 14 | 14 | 4 |
Tt71: intracellular protease | 13 | 5/5 | 23/26 | 0/0 | 7/8 | 5 | NT | NT |
Tt75: prolyl endopeptidase | 29 | 18/13 | 3/0 | 5/4 | 1/5 | 15 | 11 | 1 |
Tt80: HAD-family sugar phosphatase | 31 | 17/12 | 1/0 | 0/0 | 9/6 | 24 | NT | NT |
Tt81: haloacid dehalogenase | 11 | 42/54 | 9/5 | 0/0 | 18/16 | 0 | NT | NT |
Tt82: HAD-superfamily hydrolase | 23 | 5/8 | 1/0 | 5/4 | 0/0 | 22 | 12 | 6 |
Tt94: RNA 3-terminal phosphate cyclase | 21 | 9/8 | 11/11 | 0/0 | 8/8 | 14 | NT | NT |
Tt97: aspartate racemase | 14 | 24/2 | 3/2 | 0/0 | 6/5 | 8 | NT | NT |
Tt102: endonuclease methyltransferase | 20 | 9/6 | 2/4 | 1/0 | 1/1 | 15 | 15 | 1 |
Tt106: nucleotide kinase | 16 | 5/3 | 0/0 | 0/0 | 0/0 | 15 | 14 | 4 |
Tt141: inorganic pyrophosphatase | 11 | 21/23 | 13/14 | 4/6 | 20/12 | 3 | 1 | 1 |
Tt186: alcohol dehydrogenase | 10 | 18/21 | 10/8 | 4/5 | 15/12 | 3 | NT | NT |
Tt189: nucleoside diphosphate kinase | 21 | 10/10 | 1/1 | 1/1 | 7/3 | 3 | NT | NT |
PCP: pyroglutamate aminopeptidase | 42 | 36/22 | 32/8 | 4/2 | 8/2 | 20 | 20 | 15 |
PCNA: proliferating cell nuclear antigen | 21 | 22/22 | 10/6 | 3/0 | 14/11 | 8 | NT | NT |
Phas: kidney bean phaseolin | 13 | 17/19 | 0/0 | 0/0 | 15/17 | 5 | NT | NT |
HiIPP: Haemophilus influenzae IPPase | 47 | 24/25 | 1/0 | 0/0 | 16/20 | 11 | NI | NI |
hTFN: holo transferrin | 13 | 4/6 | 0/0 | 0/2 | 2/2 | 13 | NT | NT |
BSA: bovine serum albumin | 10 | 2/2 | 1/1 | 1/0 | 0/0 | 9 | 9 | 0 |
GOL: glucose oxidase | 13 | 10/7 | 3/2 | 0/0 | 6/6 | 6 | 10 | NT |
Totals | 337/295 | 137/103 | 32/25 | 156/139 | 128 | 39 |