Table 1.
CA analogs EC50 for lowering Aβ42
| ||
|---|---|---|
| R1 | Cmpd# | Aβ42 EC50 (nM) |
|
5 | 1780 |
|
6 | 1960 |
|
7 | 110 |
|
|
8 | 148 |
|
2a | 250 |
|
2b | 501 |
|
9 | 2193 |
|
10 | 391 |
|
11 | 513 |
EC50=half maximal effective concentration
CA analogs EC50 for lowering Aβ42
| ||
|---|---|---|
| R1 | Cmpd# | Aβ42 EC50 (nM) |
|
5 | 1780 |
|
6 | 1960 |
|
7 | 110 |
|
|
8 | 148 |
|
2a | 250 |
|
2b | 501 |
|
9 | 2193 |
|
10 | 391 |
|
11 | 513 |
EC50=half maximal effective concentration