Figure 3.
A) Direct ITC experiments with 2, 6 a, and 7 m against HumRADA2. B) Analysis of the thermodynamics of binding for various fragments and representative lead compounds 5 c (KD=35 μm), 6 a (KD=3 μm), and 7 m (KD=1.3 μm) to HumRADA2.
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